"Katadolon": instructions for use, price and reviews. Analog "Katadolon"

What is the drug “Katadolon”? Counterparts, and instructions for use of this medication will be represented in this article. You learn from it and how what is the remedy if there are contraindications and side effects, in which form is produced, which contains in its composition, and so on.

Package, method of production, composition

The Drug “Katadolon” goes on sale in two different forms. Their description, composition and packaging we will review right now.

• Medicine “Katadolon Forte” – biconvex yellow tablet oval shape (one side of the strip) containing various inclusions. The drug contains the active ingredient, as the maleate, flupirtine and other excipients. Tablets are placed in blisters of 10, 7 and 14 pieces, which are Packed in bundles of cardboard.
• Capsules “Katadolon Retard” in the gelatin shell is red. The content of the drug is a powder green-yellow or yellow tint. In one capsule contains the maleate flupirtine, as well as additional substances in the form of gelatin, magnesium stearate, water, titanium dioxide, E172, silicon dioxide, sodium lauryl sulfate, dihydrate calcium hydrogen phosphate and copovidone. The drug is Packed in cartons of 30, 50, or 10 capsules.

Pharmacological action of drugs

What is the drug and does he have a counterpart? “Katadolon” is a non-opioid analgesic that has anti-spastic effects, and has many different counterparts.

The Drug is not addictive and can have Central effects. After entering the body, it affects G-protein, thereby changing the potential difference in the calcium channels and stabilizing the membrane potential of neurons.

What are the properties of the drug under consideration and its counterpart? “Katadolon” should be taken in doses that do not exceed the maximum allowable. Only in this case the active substance will not affect the N - and M-cholinergic receptors, as well as opioid, dopamine, serotonin, ALPHA2 - and alpha1-adrenergic receptors.

After taking the capsules or tablets inside the pain relief is due to the opening of potassium channels that are found in the nerve cells.

According to experts, this drug has a good effect on NMDA receptors. It stops the current of calcium ions that pass through the partially permeable wall membranes.

The Principle of action drug

How the effect on the human body the tool and its counterpart? “Katadolon" contains in its composition flupirtine. This substance does not allow the nerve impulse to respond to nociceptive stimuli. As a result of such exposure is pain relief.

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The Drug does not occur pain, and also prevents them from becoming chronic. In addition, it effectively reduces existing pains.

After receiving the funds occurs inside the muscle relaxation (due to the blocking of intermediate neurons). We can not say that this drug is able to protect neurons from toxins. Activating calcium channels, the drug reduces the detrimental content of calcium ions in cells.

Pharmacokinetics of medicine

Upon receipt of the tablets and capsules “Katadolon Retard” in the digestive tract of the active substance of the medicine is completely absorbed (about 90%). With 75% of the dose is metabolized in the liver.

The half-life of the drug from the body is 7-15 hours. Up to 70% of the drug excreted by the kidneys, and the rest — by means of the bowel.

In the elderly and patients with impaired liver and kidney the half-life increases.

The Drug “Katadolon”: indications for use

Indications for use of this drug are pain of various origins (mild and moderate) that is caused by spasms of smooth muscles.

So when any deviations prescribed the tool and its counterpart? “Katadolon” is very often used for postoperative and headaches, back pain and neck malignancy and tumors, etc.

Contraindications medications

The Cure “Katadolon” it is not recommended to use in diseases of the kidneys and liver, hypoalbuminemia, Allergy to active substance or excipients, ringing in the ears, and in the treatment of the elderly, children and alcoholics.

Method of drug administration

How should I take the medication "Katadolon”? Capsules is in any case impossible to chew. The dosage of the drug chosen only on an individual basis.

In the literature accompanying the medication instructions are given the following treatment scheme:

• Adults up to 65 years appoint 100 mg four times a day (i.e. 1 capsule). You must adhere to the same intervals between doses of the drug. When expressed pain syndrome is allowed to take two capsules three times a day. It should benote that the maximum daily dose should be 600 mg (i.e., 6 capsules).
• Elderly people (after 65 years), the drug “Katadolon” should be taken at 100 mg twice a day. Depending on the degree of pain the dose can be increased to 300 mg per day.
• Patients who suffer from renal failure or hypoalbuminemia, usually no more than 300 mg per day.
• Impaired liver function the medication cannot be taken in a dose that exceeds 200 mg per day. The duration of such therapy may be different. However, long-term treatment requires monitoring of liver enzymes.

Analogues of the drug “Katadolon" contain the same active substance as the original. However, their choice as a replacement, be sure to consult a doctor and choose the optimum dosage.

Overdose medicine

There are few reports on cases of overdose “Katadolon” with suicidal intent. In this case you experience the following symptoms: nausea, a state of prostration, tachycardia, confusion, tearfulness, dry mouth, stupor.

As the treatment of such symptoms apply forced diuresis. In addition, the patient is given activated charcoal and administered electrolytes. Subject to all these measures the well-being of the patient improves after 6-12 hours.

Adverse reactions after taking the drug

Some patients after ingestion of tablets or capsules “Katadolon" can manifest side effects such as:

• Dizziness, General weakness and fatigue;
• Flatulence, nausea and abdominal pain;
• Tremor, indigestion;
• Headaches and anxiety;
• Allergic reactions;
• Drug-induced hepatitis;
• Blurred vision.

Side effects may occur suddenly and also suddenly disappear in the process of completing the course of therapy.

Drug interactions

While receiving the drug “Katadolon” such as "Warfarin" and "Diazepam" of the action of the first may increase. This is due to the fact that these medicines are easy to bind to proteins, which contributes to the displacement of flupirtine of cells.

Sedatives, muscle relaxants, and alcohol increase your effects under the influence of a drug.

Do Not combine the drug with “Often”, “Carbamazepine" and ‘Properties”.

It should Also be noted that while simultaneous use of drugs with ‘Coumarin” it is necessary to monitor the prothrombin index.

Special instructions

Before using drugs ‘Katadolon” you should read the manual. It States that:

• This drug should be used only in the case if a therapy other painkillers are contraindicated.
• During the application of the medicine in people with reduced renal function is necessary to control the concentration of creatinine in the blood.
• In patients older than 65 years and patients with hypoalbuminemia and severe renal insufficiency require dose adjustment of the drug.
• Patients need to be warned that during treatment should pay particular attention to the symptoms of liver damage. The manifestation of these signs want to stop taking the medication and consult a doctor.
• During therapy, the drug “Katadolon” possible false-positive reaction test for urobilinogen, bilirubin and protein in the urine.
• When using high doses of the drug, the patient may be urine staining in green. This is not a clinical symptom of any disease.
• During treatment it is necessary to abandon the control mechanisms and driving vehicles, as patients may develop dizziness and drowsiness.

The Drug “Katadolon”: counterparts, reviews, price

A Synonym for this tool is a drug “Flugelin”. As for analogs, these include the following medicines: “Acupan”, “Nefopam”, “Coldflu” and “Simeon”.

The drug Price considered very high. As a rule, it varies between 900-1200 rubles (depends on the shape and number of tablets, capsules).

According to the reviews of patients, the drug “Katadolon” quite effectively and quickly removes any pain. Despite the large number of adverse reactions, drug users often use this tool to pain with withdrawal.

As for regular patients, some of them complain that the reception of such medication often causes dizziness and General weakness.

According to doctors, the drug “Katadolon” is often used in surgical practice. It is a very powerful tool, so taking it without a doctor's prescription is not followed.