What is the drug “Sumatriptan”? Instructions for use of this drug, its pharmacological action, the composition and form of issue will be presented a little further. Also in this article we will tell you about what the contraindications, indications and side effects this medication has, what its methods of application and dosage, whether there are at it analogs, and so on.
Currently, the pharmacy can only find the pills and nasal spray “Sumatriptan”. Instructions for use of this tool gives full information on the composition of this drug. To see these you can right now.
The Pills in plastic shell contain such an active substance, such as sumatriptan succinate. As for support elements include: calcium hydrogen phosphate dihydrate, cellulose microcrystalline, hyprolose (or Klucel LF hydroxypropyl cellulose), magnesium stearate, mannitol (or mannitol), croscarmellose sodium (or Primerose).
Active substance nasal spray “Sumatriptan” also stands sumatriptan. As for the helpers, they can be changed in accordance with the form of release of the drug. It should be particularly noted that the spray used for the treatment of much less than pills. However, they have their consumers. As a rule, those patients who are uncomfortable taking medication oral way.
What features have tablets “Sumatriptan" reviews, which we'll explore next?
Said the drug is protivomigrenoznoe tool. It is a selective specific agonist of 5-HT1-serotonin receptors, which are localized in the blood vessels of the brain. It should be noted that the drug with no effect on other subtypes of 5-HT-serotonin receptors.
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After taking the drug it causes narrowing of the arteries belonging to the carotid arterial bed. Thus, the drug “Sumatriptan" (tablets) supplies blood intracranial and extracranial tissue. It should be noted that the expansion of blood vessels of the meninges and their swelling is the cause of development of migraine in humans.
Not to mention the fact that after the adoption of the tool has no significant effect (negative) on cerebral blood flow. Pills only suppress the activity of receptors of afferent fibers (or their endings) of the trigeminal nerve, which is located in the Dura mater. This happens due to the reduced allocation of sensory cortex.
It should Also be said that the drugs “Sumatriptan” and “Sumatriptan Teva’ eliminate photophobia, and nausea, which are directly related to migraine attacks.
As quickly comes a positive effect after the adoption of the drug “Sumatriptan”? Patients ' feedback on this drug contain information that the drug begins to act only after 30 minutes. In this case the patient must take a dose of 100 mg. by the Way, in 50-70% of cases patients rapidly eliminates migraines after using 25-100 mg of the drug. During the day in 1/3 of patients develop recurrence, which requires repeated use of the drug.
How long the drug is absorbed “Sumatriptan”? The answer to this question is also contained in the instructions for using the tool. After taking the drug inside it is almost immediately absorbed in the digestive tract. After about 45 minutes the concentration of the drug in the blood serum reaches about 70 %.
Due to incomplete absorption and first-pass metabolism the absolute bioavailability of the drug when administered on average 14 %. With regard to binding with blood plasma proteins is low (approximately 15–21 %). The half-life time is about 2 hours. The drug is excreted primarily through the kidneys.
According to experts, migraine attacks do not have a significant impact on the absorbability of the active substance sumatriptan (ingestion or intranasal administration).
If the patient has impaired function of the liver, after the use of medication it can be observed elevated levels of active ingredient in plasma. This happens as a result of lower first-pass clearance.
In any cases assigned to the drug “Sumatriptan”? Instructions for use of this drug States that it should be adopted only with the signs of the migraine attack (without aura or with it).
If there is any deviations are forbidden to take the drug “Sumatriptan”, analogs of this drug? I want to emphasize that this account of the user has a large amount of information. That is why before takingmedicines with her, be sure to see.
So what are the contraindication is represented by the drug? Consider the list right now:
As mentioned above, the drug “Sumatriptan” during pregnancy use is prohibited. But if the risk to the fetus is less than the benefit to the mother, it is still prescribed to women pregnant and nursing mothers. However, it must be done only by an experienced specialist (medication is taken strictly under his supervision). By the way, it is not recommended to breast feed the baby during the day after taking the mentioned tablets.
This drug is taken inside, regardless of meals. The dosage in this case must equal 50 mg (if necessary - 100 mg).
If you decide to use nasal medication “Sumatriptan" (spray), its dose is 20 mg in each nostril. Repeated administration of the drug allowed no earlier than 2 hours.
The Maximum daily dosage for oral administration is 300 mg. During intranasal use of the drug it is two doses of 20 mg.
Now you know how to defeat a migraine. “Sumatriptan" (tablets and spray) copes well with the task. However, it should be noted that this medication is not intended to prevent the deviation mentioned.
The Use of the drug is possible only in the case when the diagnosis is not in doubt. Before prescribing medication “Sumatriptan” for patients with atypical and not previously diagnosed with migraine, the doctor must rule out other dangerous neurological condition. You should also consider that patients referred with a diagnosis after taking the pills may develop cerebrovascular disorders.
The Presence of abnormalities in the circulatory system (for men over 40 and women post-menopausal stages) requires a preliminary examination, in order to exclude pathology of the heart and blood vessels.
Currently there is information on the onset of disorders of coordination, weakness and hyperreflexia after taking the medication “Sumatriptan” and other drugs from the group of selective inhibitors.
Before and during treatment presented by drug requires constant eating, and adhering to a strict diet. So, the patient is recommended to eliminate from your diet foods that contain the substance tyramine (chocolate, citrus, cocoa, celery, nuts, cheese, beans and tomatoes). In addition, it is necessary to abandon the use of alcoholic beverages, including red, sparkling and dry wines, champagne, beer.
Sport and healthy lifestyle in General (walking, swimming, skiing), as well as the presence of any hobby contribute to the emergence of positive emotions, which prevents the development in a human patient of migraine attacks.
Trade name of a spray with the active substance sumatriptan sounds like "Imigran". This medication has the following parts:
It Should be particularly noted that the blue button works very quickly and only once. In this regard, it is not recommended to click on it as long as the arrow will not be put in the nasal passage. Otherwise, the entire dose will be wasted.
To use the nasal spray, the patient should take a comfortable position lying down, standing or sitting. Incidentally, after the nasal cavity of the patient is recommended to be cleaned with cotton swabs.
Removing the blister pack and removing a medicament for nasal use, the drug is expected to enter into one nostril. As for the other nasal passage, it should be pressed a finger to the nasal septum. The patient must breathe through the mouth.
Insert the tip of the nasal the drug into the nostril should be 1 centimeter. The patient's head should be kept straight and not tilt back. After that, the patient should close the mouth and making quiet and slow breath through the nose, with a simultaneous effort to push the bluebutton with your thumb. With this, one can seem that the button is very tight. But it's not. In the process of injecting a medicinal substance into the nasal cavity, the patient should hear a faint clicking noise. This means that the button has successfully worked.
After this procedure the patient is required to open your mouth and slowly breathe through it. The head must continue to keep straight. Further, patients should make a quiet breath through the nasal cavity, and then exhale-through the mouth (for 10-20 seconds). It is recommended not to breathe too deeply.
After the procedure of injection of the drug is complete, the person may sense the presence of moisture in the nose and weak flavor. These sensations are not dangerous for health and very quickly they disappear. After one use, the dispenser can be discarded.
The Drug “Sumatriptan Teva" reviews, which largely are positive, you must be careful to take the drivers of vehicles, as well as those who are engaged in hazardous activities that require high-speed reactions and special attention.
Whether to trigger the emergence of side effects, the drug “Sumatriptan”? Drugs of this type can contribute to the development of a fairly large number of negative phenomena. Let's consider them in more detail:
What is the impact of other medications on the effectiveness and impact of the drug “Sumatriptan”? Manual, reviews of professionals on this score contain the following information. While using drug medication “Ergotamine” and ergotaminsoderjasimi means the patient possible long spasm. In this regard, the interval between doses of these drugs must be at least 24 hours.
According to research, there is interaction between the drug “Sumatriptan” and MAO inhibitors. Thus decreases the intensity of metabolism of the first, and increases its concentration.
While using these tools against migraine attacks and drugs belonging to the selective inhibitors of serotonin reuptake, patients may develop weakness, hyperreflexia and disrupt the coordination of movements.
What happens if you do not observe the dosage recommended by your doctor? Excessive use of the drug “Sumatriptan” in patients may increase the above adverse reactions. In this regard, their condition requires special observation for 10 hours.
If necessary, in case of overdose patient assistance in the form of symptomatic treatment.
You can Purchase this tool at any pharmacy. It should be noted that the price of the drug “Sumatriptan” compared to others, relatively low. So, for 50 tablets in plastic shell you will have to pay only 170-200 rubles. As for the nasal tools, its price is about the same.
Is There anything like drug “Sumatriptan”? “Amigrenin” is a drug which often acquire to eliminate migraines if the pharmacy absent the aforementioned means. In addition, analogues of the drug “Sumatriptan” on the active substance are the following medications: “Coumarin”, “Imigran”, “Sumatran”, “Myriam”, “Sumatriptan-Teva”, “Sumatriptan succinate”, “Sumatriptan Pfizer”, “Sumatriptan ABK”, “Sumamigren”, “Triligran” etc.
As similar to the nasal remedies some experts recommend to use a spray called "Imigran".
Presents drug should be stored only in dry protected from sunlight place. The temperature indoors should not be more than 25 degrees. Shelf life of medical devices is 3 years. After this period, the drug use is prohibited.
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Alin Trodden - author of the article, editor
"Hi, I'm Alin Trodden. I write texts, read books, and look for impressions. And I'm not bad at telling you about it. I am always happy to participate in interesting projects."
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